Selektive Herstellung einer Einzigen Axial Chiralen Verbindung

Details

Veröffentlichungs-Nr.

EP4775573

Anmeldetag

6. September 2024

Veröffentlichung

13. März 2025

Rechtsraum

EP

Abstract

The present invention, in one embodiment, relates to a method for producing a compound of formula (I) or a salt thereof, as defined in the specification. The production method includes reacting a compound of formula (IIA) or a salt thereof with a compound of formula (IIIA) or a salt thereof, or alternatively reacting a compound of formula (IIB) or a salt thereof with a compound of formula (IIIB) or a salt thereof, to obtain the compound of formula (I) or a salt thereof. In the compound of formula (I), it is preferred that R<4> is formula (VI) or (VII) and R<5> is formula (VIII) or (IX) (each of the formulas, together with R<4> and R<5>, is as defined in the specification).

Anmelder

Firma

Astellas Pharma Inc.

Land

🇯🇵 Japan